Eltrombopag 艾曲波帕; SB-497115
Eltrombopag (SB-497115),属于biarylhydrazone小分子,是一种thrombopoietin receptor (TpoR)的非肽类激动剂,用于治疗慢性丙型肝炎相关的血小板减少和慢性免疫性(自发的)血小板减少(ITP)。
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货号:
TK0567 -
规格:
- 1mg
- 10mg
- 50mg
- 100mg
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价格:
¥0.00
Eltrombopag (SB-497115),属于biarylhydrazone小分子,是一种thrombopoietin receptor (TpoR)的非肽类激动剂,用于治疗慢性丙型肝炎相关的血小板减少和慢性免疫性(自发的)血小板减少(ITP)。
| CAS No. | 496775-61-2 |
| 生物活性 | Eltrombopag (SB-497115) is a thrombopoietin (TPO) receptor agonist developed for certain conditions that lead to thrombocytopenia. |
| 分子式 | C25H22N4O4 |
| 分子量 | 442.47 |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存条件 | Powder -20°C 3 years |
| 溶解性数据 | DMSO : 8.33 mg/mL (18.83 mM; Need ultrasonic) H2O : < 0.1 mg/mL (insoluble) |
| 文献 | •Blood Adv. 2017 Feb 28;1(7):468-476. •Front Pharmacol. 2020 Nov 16;11:582625. •Viruses. 2019 Apr 25;11(4):385. •BMC Cancer. 2020 Nov 30;20(1):1171. •Curr Microbiol. 2021 Feb 21. |
| 纯度及产品资料 | 98% |