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WAY-100635 Maleate

WAY-100635 Maleate

WAY-100635 Maleate是一种有效的，选择性的5-HT1A受体拮抗剂，IC50为0.95 nM。

货号：
TK0446
规格：

1mg

5mg

10mg

50mg
价格：
￥0.00

产品参数

CAS No.	1092679-51-0
生物活性	WAY-100635 maleate is a potent and selective 5-hydroxytryptamine 1A (5-HT1A) receptor antagonist with an IC50 value of 0.91 nM and Ki value of 0.39 nM. WAY-100635 maleate has pIC50 values for 5-HT1A and α1-adrenergic receptors of 8.9 and 6.6, respectively. WAY-100635 maleate is also a potent dopamine D4 receptor agonist.
分子式	C25H34N4O2.C4H4O4
分子量	538.64
运输条件	Room temperature in continental US; may vary elsewhere.
储存条件	Powder, -20°C ,3 years
溶解性数据	DMSO : ≥ 250 mg/mL (464.13 mM),H2O : 25 mg/mL (46.41 mM; Need ultrasonic)
体内研究	WAY-100635 (1 mg/kg; subcutaneous injection; male Sprague-Dawley rats) treatment abolishes the reduction of the severity of abstinence signs induced by Rhodiola rosea administration in nicotine-dependent rat.
纯度及产品资料	98%

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