ARN-3236
ARN-3236 是一种有效的、可口服的、选择性的 salt-inducible kinase 2 (SIK2) 抑制剂，对SIK2、SIK1和SIK3的IC50值分别为 <1 nM、21.63 nM和6.63 nM。ARN-3236 在癌细胞中诱导凋亡。
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货号：
TK0422 -
规格：
- 2mg
- 5mg
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价格：
￥0.00
产品参数
| CAS No. | 1613710-01-2 |
| 生物活性 | ARN-3236 is an oral active and selective inhibitor of salt-inducible kinase 2 (SIK2), with IC50s of <1 nM, 21.63 nM and 6.63 nM for SIK2, SIK1 and SIK3, respectively. Has anti-cancer activity. |
| 分子式 | C19H16N2O2S |
| 分子量 | 336.41 |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存条件 | Powder -20°C 3 years |
| 溶解性数据 | DMSO : 100 mg/mL (297.26 mM; Need ultrasonic) |
| 体外研究 | ARN-3236 inhibits SIK2 activity with an IC50 <1 nM. ARN-3236 inhibits cell growth and increases NSC 125973 sensitivity in ovarian cancer cells. |
| 纯度及产品资料 | 98% |
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